8 research outputs found
Proteasome inhibition for treatment of leishmaniasis, Chagas disease and sleeping sickness
- Author
- AC Ivens
- Advait S. Nagle
- Agnes Biggart
- Ansgar Brock
- AP McLatchie
- Badry Bursulaya
- Ben G. Wen
- BS McGwire
- C Bern
- C Bern
- C Li
- CA Morillo
- Casey J. N. Mathison
- D Sacks
- D Steverding
- E Chatelain
- E Myburgh
- E Wirtz
- Elmarie Myburgh
- Fang Liang
- FJ Logan-Klumpler
- Frantisek Supek
- Frederick S. Buckner
- FS Buckner
- G Bilbe
- Glen Spraggon
- Glenn Federe
- H Li
- Hazel X. Y. Koh
- I Molina
- Ianne C. Rivera
- J Wang
- J. Robert Gillespie
- Jaime Ballard
- JC Kalvass
- Jeremy C. Mottram
- JM Bustamante
- Jocelyn L. Tan
- John D. Venable
- John R. Walker
- JR Coura
- JS Melnick
- KG Nelson
- Lauren C. Davis
- M Unno
- MC Nunes
- MC Taylor
- Michael Shapiro
- Monique Stinson
- Mu-Yun Gao
- NJ Waters
- NM El-Sayed
- PG Kennedy
- PJ Hotez
- Pranab K. Mishra
- R Viotti
- R Viotti
- Richard J. Glynne
- S Hariharan
- S Khare
- S Khare
- S Sundar
- S. Whitney Barnes
- Shilpi Khare
- Srinivasa P. S. Rao
- Todd Groessl
- Tove Tuntland
- TP Dorlo
- V Yardley
- Valentina Molteni
- Vince Yeh
- X Li
- Xianzhong Liu
- Y Fernandez
- Yin H. Lai
- Publication venue
- 'Springer Science and Business Media LLC'
- Publication date
- 01/01/2016
- Field of study
Chagas disease, leishmaniasis and sleeping sickness affect 20 million people worldwide and lead to more than 50,000 deaths annually. The diseases are caused by infection with the kinetoplastid parasites Trypanosoma cruzi, Leishmania spp. and Trypanosoma brucei spp., respectively. These parasites have similar biology and genomic sequence, suggesting that all three diseases could be cured with drugs that modulate the activity of a conserved parasite target. However, no such molecular targets or broad spectrum drugs have been identified to date. Here we describe a selective inhibitor of the kinetoplastid proteasome (GNF6702) with unprecedented in vivo efficacy, which cleared parasites from mice in all three models of infection. GNF6702 inhibits the kinetoplastid proteasome through a non-competitive mechanism, does not inhibit the mammalian proteasome or growth of mammalian cells, and is well-tolerated in mice. Our data provide genetic and chemical validation of the parasite proteasome as a promising therapeutic target for treatment of kinetoplastid infections, and underscore the possibility of developing a single class of drugs for these neglected diseases
Lawson Criterion for Ignition Exceeded in an Inertial Fusion Experiment
- Author
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- Acree R
- Adams J
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- Publication venue
- Publication date
- 01/01/2022
- Field of study
Lawson criterion for ignition exceeded in an inertial fusion experiment
- Author
- Abu-Shawareb H
- Acree R
- Adams J
- Adams P
- Addis B
- Aden R
- Adrian P
- Afeyan BB
- Aggleton M
- Aghaian L
- Aguirre A
- Aikens D
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- Albrecht M
- Albright BJ
- Albritton J
- Alcala J
- Alday C
- Alessi DA
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- Alfonso N
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- Ali ZA
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- Amick P
- Ammula S
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- Ampleford DJ
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- Aracne-Ruddle C
- Araya E
- Arend M
- Arnold P
- Arnold T
- Asay J
- Atherton LJ
- Atkinson D
- Atkinson R
- Auerbach JM
- Austin B
- Auyang L
- Awwal AS
- Ayers J
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- Azevedo S
- Bachmann B
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- Bailey DS
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- Bass I
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- Baxamusa SH
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- Benage JF
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- Besenbruch G
- Betcher J
- Bettenhausen R
- Betti R
- Bezzerides B
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- Publication venue
- 'American Physical Society (APS)'
- Publication date
- 06/07/2022
- Field of study
For more than half a century, researchers around the world have been engaged in attempts to achieve fusion ignition as a proof of principle of various fusion concepts. Following the Lawson criterion, an ignited plasma is one where the fusion heating power is high enough to overcome all the physical processes that cool the fusion plasma, creating a positive thermodynamic feedback loop with rapidly increasing temperature. In inertially confined fusion, ignition is a state where the fusion plasma can begin "burn propagation" into surrounding cold fuel, enabling the possibility of high energy gain. While "scientific breakeven" (i.e., unity target gain) has not yet been achieved (here target gain is 0.72, 1.37Â MJ of fusion for 1.92Â MJ of laser energy), this Letter reports the first controlled fusion experiment, using laser indirect drive, on the National Ignition Facility to produce capsule gain (here 5.8) and reach ignition by nine different formulations of the Lawson criterion
Prolonged expression of lipopolysaccharide (LPS)-induced inflammatory genes in whole blood requires continual exposure to LPS
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Lawson Criterion for Ignition Exceeded in an Inertial Fusion Experiment
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- Publication venue
- 'American Physical Society (APS)'
- Publication date
- 01/01/2022
- Field of study
Lawson Criterion for Ignition Exceeded in an Inertial Fusion Experiment
- Author
- Abu-Shawareb H
- Acree R
- Adams J
- Adams P
- Addis B
- Aden R
- Adrian P
- Afeyan B
- Aggleton M
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- Publication venue
- Publication date
- 01/01/2022
- Field of study
Recent Developments in Drug Discovery for Leishmaniasis and Human African Trypanosomiasis
- Author
- Advait S. Nagle
- Ahluwalia S.
- al-Gindan Y.
- Albert M. A.
- Alexandrino-de-Oliveira P.
- Alp M.
- Alrajhi A. A.
- Alvar J.
- Alvar J.
- Amaro R. E.
- Anabwani G. M.
- Andriy Buchynskyy
- Ankisetty S.
- Aponte J. C.
- Arafa R. K.
- Arana B. A.
- Armijos R. X.
- Arun Babu Kumar
- Ashburn T. T.
- Attar Z. J.
- Baiocco P.
- Bakuna S. M.
- Bakunov S. A.
- Bakunova S. M.
- Balana-Fouce R.
- Balana-Fouce R.
- Barea C.
- Barrett M. P.
- Becker I.
- Belehu A.
- Ben Achour Y.
- Ben Salah A.
- Benson T. J.
- Berg M.
- Berman J.
- Berman J. D.
- Bern C.
- Bernardes L. S.
- Bhandari K.
- Bhattacharya S.
- Bincoletto C.
- Blum J.
- Boitz J. M.
- Bolognesi M. L.
- Borges A.
- Bowyer P. W.
- Brahmachari U. N.
- Brand S.
- Brannigan J. A.
- Brenzan M. A.
- Brenzan M. A.
- Brenzan M. A.
- Breuning A.
- Brown M.
- Brun R.
- Brun R.
- Brustoloni Y. M.
- Caffrey C. R.
- Calogeropoulou T.
- Calvopina M.
- Campos S. M.
- Capewell P.
- Carballeira N. M.
- Carballeira N. M.
- Carballeira N. M.
- Carballeira N. M.
- Carballeira N. M.
- Carvalho L.
- Casey J. N. Mathison
- Cavalli A.
- Cavalli A.
- Cavazzuti A.
- Chakravarty J.
- Chan M. M.
- Chan M. M.
- Chandra S.
- Changtam C.
- Chappuis F.
- Chauhan K.
- Chawla B.
- Checchi F.
- Choe J.
- Chowdhury S.
- Chudzik D. M.
- Chulay J. D.
- Chulay J. D.
- Chunge C. N.
- Cleghorn L. A. T.
- Coimbra E. S.
- Colotti G.
- Colotti G.
- Cook G. C.
- Cordeiro A. T.
- Cordeiro A. T.
- Corona P.
- Cotterell S. E.
- Cragg G. M.
- Croft S. L.
- Cui L.
- Cunha A. M.
- Cunha R. L.
- Cunha R. L. O. R.
- da Silva L. E.
- da Silva L. E.
- Das A.
- Das B. B.
- Das B. B.
- Das P.
- Datta R.
- Davidson R. N.
- De Muylder G.
- de Oliveira A. M.
- De Rycker M.
- de Souza Pietra R. C.
- Delgado J.
- Desjeux P.
- Di Cristina G.
- Diaz-Gonzalez R.
- Ding D.
- Doerig C.
- Dorlo T. P.
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- Duarte N.
- Duncan R.
- Dye C.
- Edwards D. I.
- Edwards D. I.
- Eissa M. M.
- Ejazi S. A.
- Enanga B.
- Endeshaw M.
- Esfandiarpour I.
- Fairlamb A. H.
- Ferreira M. E.
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- Fevre E. M.
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- Foroumadi A.
- Foroumadi A.
- Foulet F.
- Franke E. D.
- Frantisek Supek
- Frederick S. Buckner
- Freire M.
- French J. B.
- Fricker S. P.
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- Fulwiler A. L.
- Furtado T. A.
- Fyfe P. K.
- Fyfe P. K.
- Galiana-Rosello C.
- Gazanion E.
- George T. G.
- Georgopoulou K.
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- Gibson W. C.
- Giri O. P.
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- Gontijo V. S.
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- Guillon J.
- Gul W.
- Hailu A.
- Hardy L. W.
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- Hemsworth G. R.
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- Hurissa Z.
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- Ishigami S. T.
- Jacobs R. T.
- Jarvis J. N.
- Jean-Moreno V.
- Jha S. N.
- Johner A.
- Kaiser M.
- Kato N.
- Kedzierski L.
- Kedzierski L.
- Kedzierski L.
- Kennedy P. G.
- Kerr I. D.
- Khabnadideh S.
- Khalil E. A.
- Khan M. O.
- Khandelwal K.
- Khandpur S.
- Kikuth W.
- Kossuga M. H.
- Kuhls K.
- Kumar K.
- Kumar P.
- Kumarihamy M.
- Kyriazis J. D.
- Lainson R.
- Lainson R.
- Larson E. T.
- Lawn S. D.
- Lee N.
- Lessa H. A.
- Lima C. B.
- Liotta F.
- Lizzi F.
- Llanos-Cuentas A.
- Lopez-Velez R.
- Lourie E. M.
- Lourie E. M.
- Luis L.
- Machado P. A.
- Machado P. R.
- Machumi F.
- Magaraci F.
- Mallari J. P.
- Mandal S.
- Manson-Bahr P. E. C.
- Markle W. H.
- Marsden P. D.
- Martin-Quintal Z.
- Martinez A.
- Martinez Garcia P.
- Martinez-Luis S.
- Martyn D. C.
- Matlashewski G.
- Matlashewski G.
- Matsumori N.
- Matsuo A. L.
- Matta A. A.
- Mauel J.
- McNamara C. W.
- Messori A.
- Michael H. Gelb
- Miguel D. C.
- Minodier P.
- Mishra B. B.
- Mishra B. B.
- Mishra B. B.
- Mishra J.
- Misra P.
- Mohamed-Ahmed A. H.
- Momeni A. Z.
- Momeni A. Z.
- Mondal S.
- Morgan H. P.
- Morgan R. E.
- Moskalenko N.
- Motta M. C.
- Mpamhanga C. P.
- Mueller Y.
- Mukherjee S.
- Murray H. W.
- Musa A.
- Musa A. M.
- Nagendar Pendem
- Nagle A.
- Nassiri-Kashani M.
- Naveen Kumar Chennamaneni
- Navin T. R.
- Neal R. A.
- Nicolle C.
- Nieto L.
- Nkwengoua E. T.
- Nour A. M. M.
- Novac N.
- Ochiana S. O.
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- Odonne G.
- Ogungbe I. V.
- Olin-Sandoval V.
- Oliveira J.
- Olivier M.
- Olson J. A.
- Ortega-Carnicer J.
- Paine M. F.
- Paladi Cde S.
- Paniz Mondolfi A. E.
- Papadopoulou M. V.
- Paradisi A.
- Parsons M.
- Patel T. A.
- Patrick D. A.
- Patrick D. A.
- Patterson S.
- Pavli A.
- Payne D. J.
- Pearson R. D.
- Pereira I. O.
- Perry M. R.
- Plimmer H. G.
- Polonio T.
- Poorrajab F.
- Porcheddu A.
- Prata A.
- Priotto G.
- Priotto G.
- Rahman A. A.
- Rahman A. A.
- Ramesh V.
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- Rangel H.
- Rapp C.
- Reichwald C.
- Reynolds K. A.
- Riente R. R.
- Ritmeijer K.
- Ritmeijer K.
- Ritmeijer K.
- Rocha L. G.
- Rodrigues R. F.
- Rodrigues R. F.
- Roldos V.
- Rosenthal E.
- Rosenthal E.
- Rotella D. P.
- Roussel M.
- Ryczak J.
- Sacks D. L.
- Saenz R. E.
- Saenz R. E.
- Saha P.
- Saha S.
- Salerno Pimentel I. A.
- Salih N. A.
- Sanders J. M.
- Sands M.
- Saravia N. G.
- Savai R.
- Schmid C.
- Schmidt T. J.
- Schmidt T. J.
- Schroder J.
- Seaman J.
- Seebeck T.
- Seligmann J.
- Selzer P. M.
- Sen R.
- Shakur Y.
- Shakya N.
- Shalev M.
- Sharlow E. R.
- Sharma M.
- Shen T.
- Shi W.
- Shilpi Khare
- Silva C.
- Simarro P. P.
- Simarro P. P.
- Singh M.
- Singh S.
- Sinha P. K.
- Siqueira-Neto J. L.
- Siqueira-Neto J. L.
- Sobarzo-Sanchez E.
- Solomon M.
- Solomon M.
- Sousa Ade Q.
- Souza T. A.
- Stec J.
- Steert K.
- Steverding D.
- Sundar S.
- Sundar S.
- Sundar S.
- Sundar S.
- Sundar S.
- Sundar S.
- Sundar S.
- Sundar S.
- Sundar S.
- Suryawanshi S. N.
- Suzuki E.
- Swenerton R. K.
- Swinney D. C.
- Swinney D. C.
- Tahghighi A.
- Tahghighi A.
- Takasu K.
- Tarral A. B. S.
- Tatipaka H. B.
- Tatipaka H. B.
- Tempone A. G.
- ter Horst R.
- Thakur C. P.
- Thakur C. P.
- Thakur C. P.
- Thakur C. P.
- Tipparaju S. K.
- Tiuman T. S.
- Tiuman T. S.
- Tolomeo M.
- Torreele E.
- Torres-Gomez H.
- Trudel N.
- Tuntiwechapikul W.
- ul Bari A.
- Urbina J. A.
- Valentina Molteni
- van der Peet P.
- van Griensven J.
- Van Voorhis W. C.
- Verma S.
- Vianna G.
- Vianna G.
- Vicens Q.
- Vickers T. J.
- Vik A.
- Vincent I. M.
- Walker R. G.
- Wang H.
- Weina P. J.
- Werbovetz K. A.
- White R. E.
- Wiese M.
- Wilcocks C.
- Wong I. L. K.
- World health organization
- Wyllie S.
- Wyllie S.
- Wyllie S.
- Yang M.
- Yau W. L.
- Zhu X.
- Zijlstra E. E.
- Zijlstra E. E.
- Zilberstein D.
- Publication venue
- 'American Chemical Society (ACS)'
- Publication date
- Field of study
SCF-KIT signaling induces endothelin-3 synthesis and secretion: Thereby activates and regulates endothelin-B-receptor for generating temporally- and spatially-precise nitric oxide to modulate SCF- and or KIT-expressing cell functions
- Author
- A Aicher
- A Barlow
- A Bouallegue
- A Contestabile
- A Inoue
- A Jezierski
- A Namiki
- A Owada
- A Quintás-Cardama
- A Schuh
- A Tefferi
- A Tefferi
- AG Baynash
- AJ Bagnall
- AP Davenport
- Arnie Jimenez
- AS Di Nunzio
- B Heissig
- Benjamin K. Chan
- BJ Kim
- C Boulanger
- C Kalka
- C Lameu
- C Morgazo
- C Roméro-Graillet
- CD Mol
- CH Hu
- Chongjuan Wei
- CR Bacon
- CR Tirapelli
- CY Ni
- D Luque Contreras
- D Tousoulis
- DE Williams
- DP Casey
- DR Seals
- E Bernal-Mizrachi
- E Buchdunger
- E Deliu
- E Weisberg
- EA Coon
- EJ Dickson
- F Desjardins
- F Mori
- G Ari
- G Gugliotta
- G Kapakos
- G Perfume
- G Perfume
- G Sommer
- G Yetik-Anacak
- George M. Rodgers
- GM Ellison
- H Maeda
- H Yoshida
- HO Lee
- HR Chang
- HY Lin
- I Anita
- J Emole
- J Hasegawa
- J Herrmann
- J Herrmann
- J Li
- J Liang
- JA Holden
- JD Wood
- Jing Zhu
- JJ Yohn
- JM Grichnik
- Jonathan Schumacher
- K Bantubungi
- K Haglund
- K Hebeiss
- K Mujoo
- K Yamada
- KJ Aichberger
- L Levato
- L Rönnstrand
- L Sobrevia
- Latha Ramdas
- Launce Gouw
- Lei L. Chen
- Liansheng Zhang
- LL Chen
- LL Chen
- M Amyere
- M Brand
- M Ii
- M Ito
- M Krishnamurthy
- M Miettinen
- M Okura
- M Picardo
- M Yanagisawa
- Marco A. Velasco
- Marsha L. Frazier
- MD Herrera
- Michael Bader
- MQ Mazzuca
- MQ Mazzuca
- MQ Mazzuca
- MS Jaureguiberry
- MT Aye
- N Fukuda
- NP Agaram
- OA Al-Shboul
- P Anversa
- P Blume-Jensen
- P Dentelli
- P Le Coutre
- P Rajendran
- P Valent
- Pamela B. Cassidy
- PJ Kuhlencordt
- PO Bayguinov
- PW Manley
- PW Manley
- PW Manley
- R Balez
- R Lees-Green
- R Roskoski Jr
- R Weller
- R Weller
- RA Larson
- RF Furchgott
- RJ Garcia
- Robert H. I. Andtbacka
- Robert S. Benjamin
- RP Brandes
- RR Magness
- S Hori
- S Iino
- S Ishii
- S Kohgami
- S McIlhenny
- S Moncada
- S Ro
- S Torihashi
- S Verma
- Sancy A. Leachman
- Sheryl R. Tripp
- SJ Hwang
- SR McLean
- T Emori
- T Ikuta
- T Kristensen
- T Kunisada
- T Lattmann
- T Mirault
- T Quaschning
- T Walsh
- TD Kim
- U Giri
- V Gil
- V Munugalavadla
- VC Broudy
- Victor G. Prieto
- W Choi
- W Tong
- W Zhong
- Y Hirata
- Y Kawaguchi
- Y Kurohane Kaneko
- Y Mathison
- Y Mathison
- Y Ogawa
- ZC Feng
- Publication venue
- 'Public Library of Science (PLoS)'
- Publication date
- Field of study